ProName: 58786-99-5 C25H35NO8 Butorphanol tartrate
● CasNo: 58786-99-5
● Molecular Formula: C25H35NO8
● Appearance: white powder
● Application: Heterocyclic Compounds;Biochemistry;Co...
● DeliveryTime: 5-7 days after payment
● PackAge: Woven bag
● Port: whan Shanghai
● ProductionCapacity: 2 Kilogram/Day
● Purity: 99%
● Storage: Normal temperature
● Transportation: Ocean shipping Express delivery
● LimitNum: 15 Gram
butorphanol tartrate basic information
morphinan-3,14-diol, 17-(cyclobutylmethyl)-, (s-(r*,r*))-2,3-dihydroxybutanedioate (1:1) (salt);morphinan-3,14-diol, 17-(cyclobutylmethyl)-,(s-(r,r))-2,3-dihydroxybutanedioate (1:1) (salt);morphinan-3,14-diol,17-(cyclobutylmethyl)-,(s-(r*,r*))-2,3-dihydroxybutanedi;oate(1:1)(salt);stadol;torate;torbutrol;butorphanol tartrate
butorphanol tartrate chemical properties
cas database reference
58786-99-5(cas database reference)
Bhutto butorphanol tartrate
Opioid receptor butorphanol tartrate Bhutto main metabolites of excited K-, with dual agonist or antagonist of U- receptor.It is mainly with the central nervous system (CNS) in the indirect interaction between these receptors play its pharmacological effects including analgesic effect. In addition to the analgesic effect and influence on CNS including reduced respiration, spontaneous respiratory cough, vomiting, miosis, excited central sedative pharmacological effects. The effect may be achieved through non CNS mechanism. Such as the change of cardiovascular (nerve) resistance and capacitance, bronchomotor tone and gastrointestinal secretion activity of smooth muscle and bladder sphincter activity.
Chinese name Butorphanol Tartrate Injection
English name Butorphanol Tartrate Injection
Brand name Dahua
The main component Bhutto butorphanol tartrate
The name of the drug
Generic name: Butorphanol Tartrate Injection
[Jiushisuan Butuofeinuo Zhusheye]: Chinese Pinyin
[main ingredients] this product is mainly composed of: tartaric acid Bhutto butorphanol, chemical name: L - (-) -17- ring -3,14- two hydroxy butyl methyl morphine Nang D- (-) - tartaric acid (1:1) salt.
[type] central analgesic drugs
[molecular formula]: C21H29NO2 - C4H6O6
Molecular weight: 477.56 
[properties] this product is a colorless and transparent liquid
[packing] brown bottle, 5 bottles / box.
pharmacology and toxicology
The analgesic effect of general intravenous injection of a few minutes, to 10-15 minutes of intramuscular injection.Intravenous injection, intramuscular injection for 30-60 minutes and reached the peak, maintenance time is 3-4 hours, and meperidine and pentazocine, morphine.
This product can quickly reach the intramuscular absorption, peak plasma concentration in 20-40 minutes. The serum protein binding rate is about 80%, and in a concentration dependent manner in the concentration range of not more than 7ng/ml in. This product can pass through the blood-brain barrier and the placenta barrier, can enter the milk, mainly in the liver metabolism, the main metabolites were hydroxylated Bhutto butorphanol. Renal dysfunction creatinine clearance < 30 ml / min, the half-life is about 10.5 hours, the elimination rate of body fluids is 150L/H. 70%-80% drugs through urine elimination, only 15% by fecal elimination.